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CAY10471 Racemate

CAS No. 844639-57-2

CAY10471 Racemate( TM30089 Racemate )

Catalog No. M20762 CAS No. 844639-57-2

CAY 10471 is a potent highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the human CRTH2/DP2 DP1 and TP receptors( Ki values of 0.6 1200 and >10000 nMrespectively).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CAY10471 Racemate
  • Note
    Research use only, not for human use.
  • Brief Description
    CAY 10471 is a potent highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the human CRTH2/DP2 DP1 and TP receptors( Ki values of 0.6 1200 and >10000 nMrespectively).
  • Description
    CAY 10471 is a potent highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the human CRTH2/DP2 DP1 and TP receptors( Ki values of 0.6 1200 and >10000 nMrespectively).
  • In Vitro
    CAY10471 Racemate (Compound 13) inhibits PGD2-induced inositol phosphate or cAMP formation, suppresses β-arrestin translocation with IC50s of 12 and 3 nM, respectively.
  • In Vivo
    ——
  • Synonyms
    TM30089 Racemate
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    GPR
  • Recptor
    CRTh2 (DP2) receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    844639-57-2
  • Formula Weight
    416.47
  • Molecular Formula
    C21H21FN2O4S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:150 mg/mL (360.17 mM)
  • SMILES
    CN(C1CCc2c(C1)c1ccccc1n2CC(O)=O)S(=O)(=O)c1ccc(F)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ulven T Kostenis E . Minor Structural Modifications Convert the Dual TP/CRTH2 Antagonist Ramatroban into a Highly Selective and Potent CRTH2 Antagonist[J]. Journal of Medicinal Chemistry 2005 48(4):897-900.
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